Table 2 -.
Anakinra | Rilonacept | Canakinumab | |
---|---|---|---|
Pharmacology | IL-1 receptor antagonist | IL-1 receptor fusion protein | IL-1β monoclonal antibody |
Half- life | ~4–6 hours | ~8 days | ~26 days |
Approved Dosage (Ped) | 100 mg (1–8 mg/kg) sq | 160–320 mg (2.2–4.4 mg/kg) sq | 150 – 300 mg (2–4 mg/kg) sq |
Dosage Frequency | 1 day | 1 week | 4–8 weeks |
Side Effects | Infection, site reaction | Infection, site reaction | Infection, vertigo |
FDA approval (Age) | CINCA/NOMID (8 mo) | FCAS / MWS (12 yrs) | FCAS / MWS (2 yrs) |
EMA approval (Age) | CAPS (8 mo) | CAPS (2 yrs) |
Cryopyrin associated periodic syndrome (CAPS), Familial cold autoinflammatory syndrome (FCAS), Muckle-Wells syndrome (MWS), Chronic infantile neurologic cutaneous articular (CINCA) syndrome or Neonatal onset multisystemic inflammatory disease (NOMID), Pediatric dosing (Ped), age approved for treatment (Age), milligram (mg), kilogram (kg), subcutaneous (sq).