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. 2021 Nov 11;29(2):449–467. doi: 10.1007/s40199-021-00422-8

Table 4.

Categories of drugs in registered RCTs

Drugs’ category Number
Antimalarials 198

• HCQ or CQ

• artesunate

• artemisinin

• mefloquine

185

5

4

2

Antibiotics / Antifungals 100

• azithromycin

• doxycycline

• co-trimoxazole

• itraconazole

• clarithromycin

68

15

4

3

3

Glucocorticoids 108

• dexamethasone

• methylprednisolone

• budesonide

• ciclesonide

• prednisolone

• prednisone

34

31

10

10

7

6

Immunoglobulins and monoclonal antibodies 143

• IVIG

• bamlanivimab

• clazakizumab

• casirivimab + imdevimab

• bevacizumab

• mavrilimumab

24

13

6

6

4

3

Antihypertensive agents 72

• losartan

• ACE-inh

18

9

Mucolytics 36

• NAC

• dornase alfa

• bromhexine hydrochloride

18

13

10

Anticoagulants /Antiplatelets 128

• heparin

• enoxaparin

• aspirin

• nafamostat mesylate

• rivaroxaban

• dipyridamole

29

26

15

10

10

3

Hormones 33

• melatonin

• thymosin

• estradiol

• liothyronine

• oxytocin

14

7

3

2

1

Other synthetic drugs 318

• colchicine

• atorvastatin

• surfactant

• famotidine

• pirfenidone

• isotretinoin

• deferoxamine

• aviptadil

38

14

8

7

7

6

4

3

Stem cell therapies 103
Antivirals 315

favipiravir

LPV/r

remdesivir

sofosbuvir + daclatasvir

umifenovir

ribavirin

oseltamivir

molnupiravir

sofosbuvir + ledipasvir

ASC09

azvudine

71

62

39

24

18

8

7

6

6

5

4

Other Antiparasitics 140

ivermectin

nitazoxanide

niclosamide

92

24

19

Immunomodulators 287

tocilizumab

IFNs

anakinra

baricitinib

sarilumab

cyclosporine

leflunomide

interleukin-7

sirolimus

adalimumab

67

49

22

14

11

10

8

6

6

6

Antineoplastic agents 112

ruxolitinib

acalabrutinib

imatinib

tofacitinib

lenzilumab

ibrutinib

19

7

6

5

4

4

Antihyperglycemic agents 21

pioglitazone

linagliptin

metformin

4

3

5

Antifibrinolytics 42

camostat mesylate

ulinastat

tranexamic acid

29

4

3

Mineral/Vitamins 172

vitamin C

vitamin D3

zinc

vitamin A

48

45

27

9

Other biologic interventions 229
convalescent plasma 194
Vaccines 283

COVID-19 vaccine

- mRNA vaccine 71

- vector vaccines 64

- subunit vaccine 59

- inactivated vaccine 39

- DNA vaccine 13

- virus-like particle 6

- live attenuated vaccine 5

258

BCG vaccine

mycobacterium vaccine

measles vaccine

polio vaccine

6

5

3

2

*Studies may evaluate more than one intervention drug from different categories; accordingly, the sum of categories/drugs number may exceed more than 100%

Abbreviations: HCQ Hydroxychloroquine, CQ chloroquine, LPV/r lopinavir-ritonavir, IFN interferon, IVIG intravenous immunoglobulin, ACE-inh angiotensin converting enzyme inhibitors, NAC N-acetyl-cysteine, mRNA messenger ribonucleic acid, DNA deoxyribonucleic acid, BCG bacillus Calmette–Guérin