Table 2:
In vitro potency of BKI-1369 against various Cryptosporidium isolates
Cryptosporidium Isolate | EC50 (μM) |
---|---|
Cryptosporidium Production Lab Iowa C. parvum1 | 0.8 |
Bunch Grass Farm C. parvum1 | 1.1 |
C. hominis 1 | 0.3 |
Assayed using high-content imaging for Cryptosporidium proliferation: Melissa Love and Case McNamara, CALIBR/Scripps, La Jolla, CA, adapted from data in (Hulverson et al., 2017a)