Table 1.
CYP3A4 Inhibitors | CYP2C9 Inhibitors | OATP1B1 Inhibitors | Glucuronidation Inhibitors |
---|---|---|---|
Protease inhibitors Macrolide antibiotics Azole antifungals Non-dihydropyridine calcium channel blockers (diltiazem and verapamil) Antidepressants (nefazodone) Cyclosporine Amiodarone Drinking large amounts of grapefruit juice or cranberry juice (N250 mL per day) |
Fluconazole Amiodarone Fenofibrate (mild-to-moderate effect) |
Cyclosporine Protease inhibitors |
Gemfibrozil |