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. 2021 Oct 23;17:191–203. doi: 10.1016/j.ijpddr.2021.10.002

Table 1.

IC50 (μM) values for P-glycoprotein inhibitors and macrocyclic lactones for the inhibition of Tca-Pgp-11.1 as measured by H3342 efflux assays.

Drugs IC50 95% CI
Verapamil 3.32 μM 1.16 μM – 10.37 μM
Valspodar 3.01 μM 0.43 μM – 21.75 μM
Tariquidar 68.46 μM 4.13 μM–217.9 μM
Ivermectin 321.5 μM 282.7 μM–805.1 μM
Selamectin 1024.5 μM 551.8 μM – 3173 μM
Moxidectin Not Determined Not Determined