Table 1.
IC50 (μM) values for P-glycoprotein inhibitors and macrocyclic lactones for the inhibition of Tca-Pgp-11.1 as measured by H3342 efflux assays.
Drugs | IC50 | 95% CI |
---|---|---|
Verapamil | 3.32 μM | 1.16 μM – 10.37 μM |
Valspodar | 3.01 μM | 0.43 μM – 21.75 μM |
Tariquidar | 68.46 μM | 4.13 μM–217.9 μM |
Ivermectin | 321.5 μM | 282.7 μM–805.1 μM |
Selamectin | 1024.5 μM | 551.8 μM – 3173 μM |
Moxidectin | Not Determined | Not Determined |