Table 1.
Structures, cLogP Values, and Antimycobacterial Minimum Inhibitory Concentration (MIC) Values of Series 1–6 Compounds on M. bovis Bacillus Calmette-Guerin (BCG)
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Minimum inhibitory concentration required to reduce growth by 90% compared to untreated controls. Mean (±SD) of n = 3 separate determinations. For n = 2, the value of each determination is indicated. MIC90’s of clofazimine and isoniazid (INH) were 0.40 and 3.2 μM, respectively.
cLogP is an estimate of lipophilicity, and values were determined using ChemDraw Professional Version 15.1.0.144.