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Dissociation constants, Ki (μM) ± SE, for reversible inhibition of human acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) with new oximes at 25 °C.
| Thienostilbene Oximes | AChE | BChE |
|---|---|---|
| trans,syn-13 | 46 ± 7 | 355 ± 26 |
| trans,anti-13 | 41 ± 4 | 322 ± 38 |
| trans,syn-14 | 67 ± 12 | 271 ± 24 |
| trans,anti-14 | 54 ± 7 | 172 ± 14 |
| trans,syn-15 | 52 ± 12 | 573 ± 35 |
| trans,anti-15 | 76 ± 21 | 482 ± 45 |
| trans,anti-16 | 158 ± 40 | 44 ± 9 |
| cis,syn-18 | 39 ± 11 | 89 ± 16 |
