Table 3.

Compound 20–42.

No.	Structure	Assay	Biological Data	Reference
20		LPC assay	IC50 = 5.7 nM	[62]
21		LPC assay	IC50 = 1.7 nM	[21]
22		CPF4 assay	IC50 = 1.07 μM
23		LPC assay	IC50 = 28 nM
24		TG-mTMP assay	IC50 = 180 nM	[65]
25		TG-mTMP assay	IC50 = 580 nM
26		TG-mTMP assay	IC50 = 13 nM
27		TG-mTMP assay	IC50 = 22 nM
28		LPC assay	IC50 = 130 nM	[66]
29		FS-3 assay	IC50 = 33.8 nM	CN107266356
30		FS-3 assay	IC50 = 2.19 nM	[67]
31		N.D.	N.D.
32		LPC assay Plasma assay	IC50 = 17 nM IC50 = 0.26 μM
33		LPC assay Plasma assay	IC50 = 10 nM IC50 = 55 nM
34		LPC assay	IC50 = 60 nM	[68]
35		N.D.	N.D.	[69]
36		LPC assay Plasma assay	IC50 = 2.2 nM IC50 = 29 nM	[70]
37		LPC assay Plasma assay	IC50 = 520 nM IC50 = 1070 nM	[71]
38		LPC assay Plasma assay	IC50 = 2.5 nM IC50 = 42 nM
39		LPC assay Plasma assay	IC50 ≤ 1.7 nM IC50 ≤ 2.2 nM
40		LPC assay	IC50 = 35 nM	[72]
41		LPC assay	IC50 = 800 nM
42		FS-3 assay bis-nNPP assay	IC50 = 1.23 nM IC50 = 2.18 nM	[73]