Table 3. Structure–Activity Relationships for Polar Amide Groups in the Extended Pocketb.
Solubility measurement by NMR assay.
Solubility measurement by high-performance liquid chromatography (HPLC). nc, not conducted.
Solubility measurement by NMR assay.
Solubility measurement by high-performance liquid chromatography (HPLC). nc, not conducted.