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Biochemical characterization of LSD1 inhibitors. Dose–response curves of LSD1 inhibition for tool compounds (A) and clinical stage inhibitors (B) determined with the HTRF assay. Selectivity of compounds vs other FAD-dependent enzymes (C). aValues obtained with the HTRF assay. bCompound not soluble at 100 μM. Data are represented as mean ± SD of N = 2, n = 2 or 3.
