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. 2021 Mar 24;11(20):12066–12073. doi: 10.1039/d0ra10241e

The prediction results of the 60 organic cocrystals using artificial neural network models (g cm−3 for the density units).

No. Co-formers Ref. code ρ exp ρ ANN Re%
Training dataset
1 CL-20:TNT IZUZUZ 1.911 1.930 0.994
2 CL-20:AZ2 TETTAQ 1.939 1.938 −0.052
3 CL-20:NEX-1 WEPGEG 1.882 1.874 −0.425
4 CL-2:TODAAZ HIVGAW 1.971 1.958 −0.660
5 CL-20:BQN ROSMOD 1.737 1.745 0.461
6 CL-20:DNB TIVJUF 1.880 1.881 0.053
7 CL-20:4,5-MDNI NILCIX 1.882 1.877 −0.266
8 HMX:PNO WEPTAP 1.700 1.697 −0.176
9 HMX:FA ZEZHET 1.687 1.687 0
10 BTF:TNA ZEVNUL 1.811 1.819 0.442
11 BTF:MATNB GEXMON 1.804 1.814 0.554
12 BTF:TNA GEXMIH 1.884 1.867 −0.902
13 TNT:NNAP TOZMUS 1.539 1.565 1.689
14 TNT:1-BN URIJAH 1.737 1.698 −2.245
15 TNT:Ant URIJEL 1.515 1.532 1.122
16 TNT:9-BN URIJIP 1.688 1.715 1.600
17 TNT:Per URIJUB 1.531 1.536 0.327
18 TNT:T2 URIKEM 1.677 1.675 −0.119
19 TNT:DMB URILEN 1.501 1.508 0.466
20 ABA:TNT URILUD 1.594 1.589 −0.314
21 MACIC:TZM ACERAD 1.605 1.623 1.121
22 MBD:MTNB DIFZOK 1.522 1.480 −2.760
23 PM:UREA EFOZAB03 1.644 1.648 0.243
24 MC:PC FIXROV01 1.606 1.661 3.425
25 NDT:THTZT FOYSUJ 1.664 1.657 −0.421
26 IDT:NTZ FUFSOQ 1.644 1.651 0.426
27 DNBA:BA GAUTAM15 1.697 1.655 −2.475
28 PZ:OA GUDSUV 1.609 1.627 1.119
29 TNP:MDNI HARJOB 1.769 1.768 −0.057
30 NF:CA LEWTAK 1.627 1.627 0
31 NF:UREA ORUXUV 1.661 1.652 −0.542
32 NPO:PA OWIYEZ 1.682 1.653 −1.724
33 UREA:CA PANVUV 1.672 1.654 −1.077
34 PZCX:DHXBED PAQNOM 1.628 1.608 −1.229
35 DNPA:ODADA QARQUY 1.775 1.772 −0.169
36 TNP:TAD QONYUP 1.685 1.655 −1.780
37 IZO:DLTA RUWPEG 1.656 1.648 −0.483
38 IZO:LTA UHACIQ 1.631 1.646 0.920
39 IZO:LTA UHAFEP 1.607 1.616 0.560
40 DNBZA:TZ UNAWUD 1.640 1.655 0.915
41 TZTM:HP YAFFUJ 1.636 1.635 −0.061
42 BM:TNP YUQHEY 1.616 1.663 2.908
Test dataset
43 CL-20:MTNP QAPNAZ 1.932 1.928 −0.207
44 CL-20:GTA XAQFUS 1.650 1.571 −4.788
45 CL-20:NFQN ROSMIX 1.774 1.659 −6.483
46 DHDS:TZM ACETEJ 1.625 1.655 1.846
47 AB:MTNB FONHOH 1.442 1.513 4.924
48 DNBA:TA IJAKAH 1.635 1.655 1.223
49 NMI:NMI ITIXUE 1.660 1.657 −0.181
50 AN:HP JOZZED 1.614 1.647 2.045
51 Urea:OA UROXAM 1.679 1.605 −4.407
Validation dataset
52 CL-20:DNG JABYOD 1.750 1.770 1.143
53 HMX:PDCA ZEZGOC 1.630 1.658 1.718
54 BTF:TNB GEXMED 1.806 1.838 1.772
55 TNT:DMDBT URIKUC 1.496 1.523 1.805
56 TNT:PDA URILAJ 1.578 1.561 −1.077
57 TNT:TNB NIBJUF 1.640 1.653 0.793
58 DNBZA:NA AWUDEB 1.607 1.671 3.983
59 PZCX:OA UZODUK 1.628 1.651 1.413
60 TZA:NDTZI VAZBIJ 1.790 1.698 −5.140