Skip to main content
. 2021 Dec 16;13(12):2171. doi: 10.3390/pharmaceutics13122171
AUC area under the plasma concentration—time curve
AUCinf area under the plasma concentration—time curve from dosing to infinity
AUClast area under the plasma concentration—time curve from dosing to the time of the last measured plasma concentration
Cmax maximal plasma concentration
Ct trough plasma concentration
C12 plasma concentration at 12 h after administration
C24 plasma concentration at 24 h after administration
tmax time to maximal plasma concentration
t 1/2 elimination half-life
S.D. standard deviation
C.V. coefficient of variation
AE adverse event
mCRPC metastatic castration resistant prostate cancer
mCSPC metastatic castration sensitive prostate cancer
FDA Food and Drug Administration
PSA prostate specific antigen
PFS progression free survival
SGF simulated gastric fluid
FaSSIF fasted state simulated intestinal fluid
ECG electrocardiogram
QD once daily
GMR geometric mean ratio
LC liquid chromatography
MS mass spectrometry
TOS tablet for oral suspension
R-AA reference abiraterone acetate