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. 2021 Nov 30;64(24):17901–17919. doi: 10.1021/acs.jmedchem.1c01212

Scheme 2. Reagents and Conditions: (a) NaH (60% Dispersion in Mineral Oil), 0 °C, DMF then 4 h, rt; (b) ACy (i–viii), K2CO3 (1.1 equiv), NaI (1.1 equiv), CH3CN, Reflux, 3 h.

Scheme 2