Table 2.
N (%) | Selinexor 60 mg QW/BIW + carboplatin 6 AUC Q3W (N = 6) | Selinexor 60 mg QW/BIW + doxorubicin 60 mg/m2 + cyclophosphamide 600 mg/m2 Q3W (N = 4) | Selinexor 40 mg QW + FOLFIRIa (N = 3) | Selinexor 60 mg QW + irinotecan 125 mg/m2 D1 and 8 Q3W (N = 3) | Selinexor 40 mg QW + XELOXb (N = 3) | All patients (N = 19) | ||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|
All grades | Grade 3/4 | All grades | Grade 3/4 | All grades | Grade 3/4 | All grades | Grade 3/4 | All grades | Grade 3/4 | All grades | Grade 3/4 | |
Anemia | 5 (83) | 2 (33) | 2 (50) | 0 | 1 (33) | 0 | 1 (33) | 0 | 1 (33) | 1 (33) | 10 (53) | 3 (16) |
Leukopenia | 4 (75) | 1 (17) | 3 (75) | 3 (75) | 3 (100) | 0 | 1 (33) | 0 | 2 (67) | 1 (33) | 13 (68) | 5 (26) |
Neutropenia | 4 (75) | 2 (33) | 3 (75) | 3 (75) | 2 (67) | 1 (33) | 2 (67) | 1 (33) | 1 (33) | 1 (33) | 12 (63) | 8 (42) |
Thrombocytopenia | 6 (100) | 3 (50) | 3 (75) | 0 | 2 (67) | 0 | 2 (67) | 0 | 3 (100) | 0 | 16 (84) | 3 (16) |
Constipation | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
Diarrhea | 2 (33) | 0 | 0 | 0 | 0 | 0 | 1 (33) | 0 | 1 (33) | 1 (33) | 4 (21) | 1 (5) |
Nausea | 4 (75) | 0 | 4 (100) | 0 | 1 (33) | 0 | 1 (33) | 0 | 3 (100) | 0 | 13 (68) | 0 |
Vomiting | 4 (75) | 0 | 3 (75) | 0 | 0 | 0 | 1 (33) | 0 | 2 (67) | 0 | 10 (53) | 0 |
Elevated AST/ALT | 0 | 0 | 0 | 0 | 1 (33) | 0 | 1 (33) | 0 | 0 | 0 | 2 (11) | 0 |
Mucositis | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
Fatigue | 4 (75) | 0 | 2 (50) | 0 | 1 (33) | 0 | 3 (100) | 1 (33) | 1 (33) | 0 | 11 (58) | 1 (5) |
Anorexia | 1 (17) | 0 | 0 | 0 | 0 | 0 | 1 (33) | 0 | 2 (67) | 0 | 4 (21) | 0 |
Hyponatremia | 3 (50) | 2 (33) | 0 | 0 | 1 (33) | 1 (33) | 1 (33) | 0 | 1 (33) | 1 (33) | 6 (32) | 4 (21) |
Hypomagnesemia | 1 (17) | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 1 (33) | 0 | 2 (11) | 0 |
Hypoalbuminemia | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
Dyspnea | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 1 (33) | 0 | 1 (5) | 0 |
Cough | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
Elevated CPK | 1 (17) | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 1 (5) | 0 |
Infection or infestation | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
Elevated lipase | 1 (17) | 1 (17) | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 1 (5) | 1 (5) |
aFOLFIRI—irinotecan of 180 mg/m2, 5-FU continuous infusion of 2400 mg/m2, 5-FU bolus of 400 mg/m2, and leucovorin of 400 mg/m2 on days 1, and 15
bXELOX—capecitabine was dosed at 900 mg/m2 orally (PO) divided into 2 doses on days 1–14, along with oxaliplatin of 130 mg/m2 IV Q3W
QW once weekly; BIW twice weekly; AUC area under curve; mg/m2 milligrams per square meter; D1 and 8 on days 1, and 8 of each cycle; Q3W every 3 weeks; ALT alanine aminotransferase; AST aspartate aminotransferase; CPK creatine phosphokinase; FOLFIRI irinotecan with fluorouracil and folinic acid; 5-FU 5-fluorouracil; XELOX capecitabine and oxaliplatin