Table 1.
Distribution of chains across human protein kinase families and conformational state labels.
| Spatial label | Dihedral label | Annotation | AGC | CAMK | CK1 | CMGC | NEK | RGC | STE | TKL | TYR | Other | Total |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DFGin | BLAminus | Active | 306 | 823 | 189 | 1187 | 0 | 0 | 216 | 401 | 545 | 172 | 3839 |
| BLBplus | SRC-inactive | 3 | 9 | 0 | 133 | 0 | 0 | 82 | 46 | 358 | 18 | 649 | |
| ABAminus | Active-like | 60 | 45 | 3 | 95 | 0 | 0 | 11 | 9 | 310 | 88 | 621 | |
| BLBminus | 0 | 7 | 0 | 121 | 1 | 0 | 19 | 18 | 54 | 10 | 230 | ||
| BLAplus | FGFR-inactive | 3 | 2 | 0 | 3 | 0 | 0 | 4 | 40 | 152 | 1 | 205 | |
| BLBtrans | CDK-inactive | 0 | 0 | 0 | 124 | 0 | 0 | 7 | 1 | 62 | 3 | 197 | |
| None | 14 | 40 | 2 | 76 | 14 | 0 | 26 | 21 | 200 | 24 | 417 | ||
| DFGinter | BABtrans | 0 | 1 | 0 | 0 | 4 | 0 | 2 | 0 | 13 | 0 | 20 | |
| None | AURKA-inactive | 10 | 69 | 0 | 15 | 2 | 0 | 7 | 4 | 32 | 0 | 139 | |
| DFGout | BBAminus | Type-2 binding | 7 | 6 | 2 | 58 | 0 | 0 | 15 | 96 | 233 | 5 | 422 |
| None | DFGout-like | 11 | 10 | 0 | 32 | 9 | 0 | 42 | 14 | 101 | 7 | 226 | |
| None | None | 7 | 43 | 0 | 87 | 19 | 0 | 17 | 2 | 32 | 5 | 212 | |
| Total | - | 421 | 1055 | 196 | 1931 | 49 | 0 | 448 | 652 | 2092 | 333 | 7177 |