Reagents and conditions: (a)631 (1) 336.2a or 336.2b, p-TSA (0.2 equiv), DCM, rt, dark, 1 h, (2) DDQ
(1 equiv), 10 min; (b)631 (1) 336.2c, CF3COOH (1 equiv), DCM, rt, dark, 90 min, (2) DDQ (2
equiv), 10 min; (c)630 (1) Pd2(dba)3, SPhos, CsF, Cs2CO3, reflux,
48 h, (2) MnO2; (d)630 NBS (0.9
equiv), CHCl3; (e)630 NBS (3.7
equiv), CHCl3; (f)630 (Bpin)2 (2.9 equiv), Pd(dppf)Cl2, KOAc, 1,4-dioxane, reflux;
(g)630 (Bpin)2 (9.8 equiv),
Pd(dppf)Cl2, KOAc, 1,4-dioxane, reflux; (h)630336.6a/336.7a (1:1),
Pd2(dba)3, PPh3, CsF, Cs2CO3, toluene/DMF, reflux, 48 h; (i)630336.6a/336.7b (1:0.5), Pd2(dba)3, PPh3, CsF, Cs2CO3, toluene/DMF, reflux, 48 h.