Table 3.
Prediction of physicochemical propertiesa of 3 and 6–31.
| Compound | miLogP | TPSA | natoms | MW | nON | nOHNH | nrotb |
|---|---|---|---|---|---|---|---|
| Standard | <5 | <140 | <500 | <10 | <5 | ≤10 | |
| 3 | 3.48 | 41.37 | 48 | 380.87 | 2 | 0 | 4 |
| 6–31 | 2.29 | 85.61 | 54 | 408.45 | 6 | 0 | 6 |
miLogP: molinspiration predicted Log P; TPSA: topological polar surface area; natoms: No. of atoms; MW: molecular weight; nON: No. of hydrogen bond acceptors; nOHNH: No. of hydrogen bond donors; nrotb: No. of rotatable bonds.