Table 3.
Excretion of MIDD0301 and its metabolites after IP injection.
| 0-24 hours | 24-48 hours | 0-48 hours | |||
|---|---|---|---|---|---|
| Feces (%)1 | Urine (%)1 | Feces (%)1 | Urine (%)1 | Feces & Urine (%)1 | |
| MIDD0301 | 43.2 ± 5.9 | 0.3 ± 0.2 | 0.3 ± 0.1 | 0.1 ± 0.04 | 43.9 ± 6.24 |
| MIDD0301 taurine | 16.2 ± 0.9 | 0.4 ± 0.1 | <LOD | <LOD | 16.6 ± 1.0 |
| MIDD0301 glucoside | <LOD | 13.9 ± 7.1 | <LOD | 2.4 ± 0.2 | 16.3 ± 7.3 |
| MIDD0301 glucuronide | <LOD | 2.8 ± 1.2 | <LOD | 0.3 ± 0.2 | 3.1 ± 1.4 |
| Total | 59.4 ± 6.8 | 17.4 ± 8.6 | 0.3 ± 0.1 | 2.8 ± 0.44 | 79.9 ± 15.94 |
% is based on moles of MIDD0301 administered; LOD, lower limit of detection; data is presented as average (n = 3) ± StD