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. 2022 Jan 3;8:792546. doi: 10.3389/fmolb.2021.792546

TABLE 3.

SOCS3 proteomimetics: name, sequence, length, and dissociation constants values (µM) toward JAK2 catalytic domain.

Name Sequence Length KD (µM)
KIR 22LKTFSSKSEYQL33 12 360 a
ESS 34VVNAVRKLQESG45 12 >>1,000 a
KIRESS 22LKTFSSKSEYQLVVNAVRKLQESG45 24 6.43 a
ESSCONG 34VVNAVRKLQESGFYWSAVT52 19 No binding
restKIRESSCONG 25FSSKSEYQLVVNAVRKLQESGFYWSAVT52 28 No binding
KIRCONG chim KβAla25FSSKSEYQL33βAlaβAla46FYWSAVT52 20 11.0 b