Table 5.
rat in vitro PPB/BHB and rat IV cassette PBL | ||||||
---|---|---|---|---|---|---|
compound number | rat PPB (fu) | rat BHB (fu) | plasma (ng/mL) | brain (ng/g) | K p | K p,uu |
(S)-17l | 0.001 | 0.001 | 30.9 | 16 | 0.52 | 0.52 |
(S)-17i | 0.004 | 0.002 | 15.7 | 37.8 | 2.41 | 1.2 |
(S)-19a | 0.022 | 0.005 | 9.21 | 20.4 | 2.22 | 0.5 |
(S)-19d | 0.017 | 0.004 | 10.9 | 46.1 | 4.23 | 1.0 |