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. Author manuscript; available in PMC: 2023 Mar 1.
Published in final edited form as: Chirality. 2021 Dec 28;34(3):521–536. doi: 10.1002/chir.23403

TABLE 2.

Reagents and conditions to functionalize the aniline nitrogen in 4-ATQs: (i) 4-ATQ derivatives (1 equiv.), N-ethyldiisopropylamine (2 equiv.), alkylbromide (1 equiv.), N,N-dimethylformamide, 70 °C, 24h; (ii) 4-ATQ derivatives (1 equiv.), alkyl isocyanate (2-3.5 equiv.), toluene (0.1 M), 80 °C, 1 day.

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