Table 2.
Compound | BBB Score | No. of HBA | No. of HBD | Molecular Weight | cLogP | PSA | No. of Rotatable Bonds | HALF-LIFE (hours) | hERG | Tox Score | Tox Groups | LD50 (mg/kg) |
---|---|---|---|---|---|---|---|---|---|---|---|---|
Analog 2 | 4.93 | 6 | 0 | 380.488 | 3.17 | 41.91 | 6 | 6.72 | 0.54 | 0 | N/A | 412 |
Donepezil | 5.28 | 5 | 0 | 379.500 | 4.46 | 32.39 | 6 | 6.72 | 0.45 | 0 | N/A | 344 |