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. Author manuscript; available in PMC: 2022 Mar 14.
Published in final edited form as: Eur J Med Chem. 2021 Dec 2;228:114011. doi: 10.1016/j.ejmech.2021.114011

Table 4.

IC50 (nM) values for TMP195 and NT160 obtained using fluorogenic assay against recombinant HDAC proteins.

# HDAC4 HDAC5 HDAC7 HDAC9 Other HDACS
TMP195 128.1 ± 13 147.9 ± 22 7.7 ± 1.2 2.4 ± 0.51 >5000
1 (NT160) 0.08 ± 0.02 1.2 ± 0.17 1.0 ± 0.2 0.9 ± 0.2 >600 ± 231