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. 2022 Apr 2;22:98. doi: 10.1186/s12906-022-03578-1

Table 2.

Inhibitory effect of Citrus extracts on the activity of NS3-NS4A. The extracts were screened using the validated FRET assay, percentage inhibition and IC50 values were calculated for each extract. The pomegranate pericarp extract was used as a positive control

Sr. # Scientific name Common name Plant parts used % Inhibition (a-ba*100) IC50 value (µg/mL)
1 Citrus paradisi Grapefruit Mesocarp 91% 5.79 ± 1.44
2 Citrus sinesis Orange Fruit 86% 37.19 ± 5.92
3 Citrus aurantinum Bitter Orange Fruit 85% 42.62 ± 6.89
4 Citrus reticulata Mandarin Fruit 82% 57.65 ± 3.81
5 Citrus limon Lemon Fruit 80% 66.83 ± 4.92
6 Citrus aurantinum Bitter Orange Pericarp 79% 71.94 ± 2.39
7 Citrus aurantinum Bitter Orange Mesocarp 78% 77.06 ± 4.26
8 Citrus reticulate Mandarin Seeds 77% 80.02 ± 3.67
9 Citrus sinesis Orange Seeds 75% 86.93 ± 5.16
10 Citrus reticulate Mandarin Mesocarp 74% 90.59 ± 1.89
11 Citrus paradisi Grapefruit Pericarp 71% 107.90 ± 5.64
12 Citrus paradisi Grapefruit Fruit 69% 120.30 ± 2.08
13 Citrus paradisi Grapefruit Seeds 68% 132.23 ± 2.12
14 Citrus aurantinum Bitter Orange Seeds 63% 196.40 ± 2.92
15 Punica granatum Pomegranate Pericarp 98% 5.52 ± 0.74