In vitro human plasma stability of compound 18k.
| Compd | Time point (min) | % remaining | T 1/2 (min) |
|---|---|---|---|
| 18k | 0 | 100.0 | >289.1 |
| 10 | 105.7 | ||
| 30 | 104.4 | ||
| 60 | 101.5 | ||
| 120 | 85.4 |
| Compd | Time point (min) | % remaining | T 1/2 (min) |
|---|---|---|---|
| 18k | 0 | 100.0 | >289.1 |
| 10 | 105.7 | ||
| 30 | 104.4 | ||
| 60 | 101.5 | ||
| 120 | 85.4 |