Table 2.
Oritavancin Mean (CV%) Plasma Pharmacokinetic Parameters (1200-mg Infusions)
Parameter | Current Formulation | New Formulation |
---|---|---|
Dose (mg) | 1200 | 1200 |
IV Infusion Duration | 3 hours | 1 hour |
n | 50 | 50 |
C max (µg/mL) | 112 (30.8) | 148 (29) |
T max (hour)a | 3.29 (3.02–5.83) | 1.15 (0.90–3.17) |
AUC0-72 (µg * h/mL) | 1470 (39.7) | 1460 (35.1) |
AUC0-168 (µg * h/mL) | 1760 (41.4) | 1750 (35.0) |
Abbreviations: AUC, area under the concentration-time curve; CV, coefficient of variation; IV, intravenous.
Median (minimum-maximum).