. 2020 Sep 17;3(4):742–761. doi: 10.20517/cdr.2020.45

Table 1.

Various examples of antiandrogens agents*

Antiandrogens	Mode of action
Enzalutamide	AR antagonist
Bicalutamide	AR antagonist
Ostarine	Selective AR modulator
Apalutamide	Selective and competitive inhibitor
Galeterone	CYP17 inhibitor and AR antagonist
Flutamide	AR antagonist
Cyproterone Acetate	AR antagonist
AZD3514	AR down regulator
Spironolactone	AR Antagonist
Ligandrol	Selective AR modulator
Triptophenolide	Selective AR modulator
Testolone	Selective AR modulator
EPI-001	AR N-terminal domain antagonist
Darolutamide	AR antagonist and blocks AR nuclear translocation
Dehydroepiandrosterone	AR agonist
Nilutamide	AR antagonist