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. Author manuscript; available in PMC: 2022 Apr 9.
Published in final edited form as: ACS Infect Dis. 2017 Nov 2;4(4):499–507. doi: 10.1021/acsinfecdis.7b00157

Table 5.

Antifungal activity of 17d/e against fluconazole resistant-C. albicans

Entry Strain FLUa MIC (μg/mL) MORb 17d MIC (μg/mL) 17e MIC (μg/mL)
1 SC5314 0.25 1 8 8
2 TWO7229 0.25 1 8 8
3 TWO7230 2 2 8 8
4 TWO7241 16 2, 3 8 8
5 TWO7243 128 2, 3 8 8
a

Fluconazole (FLU); data are from reference 24.

b

MOR: Mechanism of resistance; 1) None; 2) Elevated efflux pump expression; 3) Elevated ERG11 expression;