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. 2022 Mar 14;13(4):546–553. doi: 10.1021/acsmedchemlett.1c00539

Table 2. Solubility and Mouse Microsomal Stability Data.

entry compd solubilitya (μM) MLMbT1/2 (min)
1 7a 0.7 10
2 7b 0.5 10
3 7o 2.0 45
a

Kinetic solubility in aqueous PBS buffer, pH 7.4.

b

MLM = CD-1 mouse liver microsomal stability.