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. 2020 Apr 14;10(24):14337–14346. doi: 10.1039/d0ra00822b

Toxicity of anastatins A and B, and their derivatives, on PC12 cellsa.

Name IC50 (μM) Name IC50 (μM)
42a >100 38a 44.69 ± 1.38
43a >100 39a 32.82 ± 2.64
44a >100 40a 31.54 ± 0.97
42b >100 38b >100
43b >100 39b >100
44b >100 40b 53.41 ± 0.85
42c >100 38c >100
42c-1 >100 38c-1 >100
43c >100 39c >100
44c >100 40c >100
19 >100 20 >100
31 >100 30 >100
(±) Anastatins A >100 (±) Anastatins B 49.45 ± 2.03
GA >100
a

Data are presented as means ± SD.