Toxicity of anastatins A and B, and their derivatives, on PC12 cellsa.
| Name | IC50 (μM) | Name | IC50 (μM) |
|---|---|---|---|
| 42a | >100 | 38a | 44.69 ± 1.38 |
| 43a | >100 | 39a | 32.82 ± 2.64 |
| 44a | >100 | 40a | 31.54 ± 0.97 |
| 42b | >100 | 38b | >100 |
| 43b | >100 | 39b | >100 |
| 44b | >100 | 40b | 53.41 ± 0.85 |
| 42c | >100 | 38c | >100 |
| 42c-1 | >100 | 38c-1 | >100 |
| 43c | >100 | 39c | >100 |
| 44c | >100 | 40c | >100 |
| 19 | >100 | 20 | >100 |
| 31 | >100 | 30 | >100 |
| (±) Anastatins A | >100 | (±) Anastatins B | 49.45 ± 2.03 |
| GA | >100 |
Data are presented as means ± SD.