Affinity constants of positive compounds and controls.
No. | Protein name | Compound name | CAS # | k on (1/Ms) | k off (1/s) | K D (M) |
---|---|---|---|---|---|---|
1 | ELP2 | Epinephrine bitartrate | 51-42-3 | 7.83 × 102 | 5.29 × 10−4 | 6.76 × 10−7 |
2 | ELP2 | Isoprenaline hydrochloride | 51-30-9 | 9.87 × 102 | 4.54 × 10−3 | 4.60 × 10−6 |
3 | ELP2 | Gluconolactone | 90-80-2 | 2.64 × 103 | 8.19 × 10−2 | 3.10 × 10−5 |
4 | ELP2 | Temozolomide | 85622-93-1 | 1.82 × 102 | 4.62 × 10−4 | 2.53 × 10−6 |
5 | ELP2 | PLX-4720 | 918505-84-7 | 1.32 × 102 | 2.22 × 10−5 | 1.68 × 10−7 |
6 | ELP2 | RK-33 | 1070773-09-9 | 5.38 × 101 | 2.59 × 10−5 | 4.81 × 10−7 |
7 | ELP2 | 5-Hydroxymethyl tolterodine | 207679-81-0 | 1.13 × 104 | 1.66 × 10−2 | 1.47 × 10−6 |
Blank | ELP2 | DMSO (solvent) | 67-68-5 | 1.71 × 100 | 7.40 × 10−1 | 4.32 × 10−1 |