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. 2019 Jan 14;9(3):1696–1704. doi: 10.1039/c8ra09640f

Affinity constants of positive compounds and controls.

No. Protein name Compound name CAS # k on (1/Ms) k off (1/s) K D (M)
1 ELP2 Epinephrine bitartrate 51-42-3 7.83 × 102 5.29 × 10−4 6.76 × 10−7
2 ELP2 Isoprenaline hydrochloride 51-30-9 9.87 × 102 4.54 × 10−3 4.60 × 10−6
3 ELP2 Gluconolactone 90-80-2 2.64 × 103 8.19 × 10−2 3.10 × 10−5
4 ELP2 Temozolomide 85622-93-1 1.82 × 102 4.62 × 10−4 2.53 × 10−6
5 ELP2 PLX-4720 918505-84-7 1.32 × 102 2.22 × 10−5 1.68 × 10−7
6 ELP2 RK-33 1070773-09-9 5.38 × 101 2.59 × 10−5 4.81 × 10−7
7 ELP2 5-Hydroxymethyl tolterodine 207679-81-0 1.13 × 104 1.66 × 10−2 1.47 × 10−6
Blank ELP2 DMSO (solvent) 67-68-5 1.71 × 100 7.40 × 10−1 4.32 × 10−1