Structures and their relative activity of DC_HG24-01 and its analoguesa.
Entry | Compound | R1 | R2 | IC50 (μM) |
---|---|---|---|---|
1 | DC_HG24 | 12.7 ± 0.9 | ||
2 | DC_HG24-01 | 3.1 ± 0.2 | ||
3 | DC_HG24-02 | 9.1 ± 1.0 | ||
4 | DC_HG24-03 | 31.3 ± 0.8 | ||
5 | DC_HG24-04 | 14.2 ± 2.1 | ||
6 | DC_HG24-05 | >100 | ||
7 | DC_HG24-06 | >100 |
Data in table is presented as mean ± SD, n = 3.