Reaction conditions and yield of products formed in S_NAr reactions of 1a with nucleophiles.

Entry	Compound	Nucleophile	Conditions	Yield [%]
1	2a	C6H5SH	TRIS, DMF, rt, 2 h	87
2	2b	4-CH3C6H4SH		89
3	2c	3,5-(CH3)2C6H3SH		81
4	2d	4-CH3OC6H4SH		95
5	2e	3-CH3OC6H4SH		84
6	2f	3-NH2C6H4SH		76
7	2g	4-BrC6H4SH		86
8	2h	C6H5CH2SH		65
9	2i	CH3(CH2)8CH2SH		37
10	2j	N-acetyl-l-cysteine methyl ester		71
11	2k	CH3NH2	DMSO, 80 °C, 3 h	71
12	2l	CH3(CH2)2NH2		74
13	2m	CH3(CH2)3NH2		60
14	2n	CH2 CHCH2NH2		65
15	2o	C6H5CH2NH2		63
16	2p	C6H5OH	K2CO3, DMF, 80 °C, 24 h	68
17	2q	4-CH3OC6H4OH		48
18	2r	4-ClC6H4OH		56
19	2s	3-NO2C6H4OH		48