Iron-catalysed alkylations of allyl acetates (condition A).
| ||||
|---|---|---|---|---|
| Entry | Allyl acetate | Product | R′ | Yielda [%] |
| 1 |
|
|
H | 85 |
| 2 | Me | 72 | ||
| 3 | nC6H13 | 67 | ||
| 4 |
|
|
61 (<5b) | |
| 5 |
|
59 | ||
| 6 |
|
|
Me | 80 |
| 7 | Cl | 0 | ||
| 8 | Br | 0 | ||
| 9 |
|
|
37c | |
| 10 |
|
|
53c | |
| 11 |
|
|
16c | |
| 12 |
|
|
64 | |
Isolated yields; E/Z product ratios >50/1.
C9H19MgCl·LiCl was used.
10 mol% Fe(OAc)2, RMgBr addition over 1 h.