Substrate scope of substituted 3,4-dihydro-2(1H)-quinazolines^a.

Entry	Substrate (2)	Amine (3)	Product (4)	Yieldb (%)
1				80
2		3a		90
3		3a		88
4		3a		85
5		3a		82
6		3a		92
7		3a		86
8		3a		70
9		3a		71
10		3a		68
11	2i			65
12	2f	3b		82
13	2h	3b		70
14	2f			80
15	2h	3c		65
16	2i	3c		66

^aUnless otherwise specified, reactions were performed using 1 equiv. of 3a, 1.2 equiv. of 2b, 3.0 equiv. of base.

^bIsolated yield.