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. 2018 Jul 11;8(44):24913–24922. doi: 10.1039/c8ra04389b

K d (μM) values for triazoles 4–9 and 12–15 and references 16–17 determined by competitive fluorescence polarization.

Galectin-1 Galectin-3 Galectin-3/galectin-1
4 370 ± 30 980 ± 60 2.6
5 120 ± 7 250 ± 20 2.1
6 61 ± 4 180 ± 10 3.0
7 47 ± 2 200 ± 10 4.3
8 47 ± 3 220 ± 10 4.7
9 140 ± 7 330 ± 20 2.4
12 58 ± 4 200 ± 7 3.4
13 43 ± 2 280 ± 7 4.5
14 62 ± 2 540 ± 30 8.7
15 180 ± 9 430 ± 20 2.4
16 1100 15 230 15 0.2
17 430 ± 40 1800 ± 100 4.2