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. 2018 Oct 22;8(63):35981–35988. doi: 10.1039/c8ra07153e

Plasma protein binding of metoprolol in BSA ( ± s, n = 3).

Drug C t (μg mL−1) C f (μg mL−1) Plasma protein binding (%)
Metoprolol 0.50 ± 0.02 0.36 ± 0.01 28.15 ± 2.02
0.99 ± 0.04 0.70 ± 0.02 29.67 ± 2.42
2.02 ± 0.06 1.45 ± 0.03 28.36 ± 1.65