IC50 Values (μM) for Nα-arylsulfonyl histamine derivatives. 1-DNJ:reference inhibitor.
| Type I compounds | IC50 (μM) |
|---|---|
| I-b | 250.00 ± 1.03 |
| I-c | 65.08 ± 1.04 |
| I-d | 79.50 ± 1.05 |
| I-e | 421.6 ± 0.94 |
| I-f | 244.2 ± 1.09 |
| I-g | 71.43 ± 1.02 |
| I-h | 72.69 ± 1.05 |
| I-i | 102.20 ± 1.05 |
| I-j | 95.55 ± 1.02 |
| 1-DNJ | 65.18 ± 1.04 |