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. 2018 Oct 24;8(63):36209–36218. doi: 10.1039/c8ra06625f

IC50 Values (μM) for Nα-arylsulfonyl histamine derivatives. 1-DNJ:reference inhibitor.

Type I compounds IC50 (μM)
I-b 250.00 ± 1.03
I-c 65.08 ± 1.04
I-d 79.50 ± 1.05
I-e 421.6 ± 0.94
I-f 244.2 ± 1.09
I-g 71.43 ± 1.02
I-h 72.69 ± 1.05
I-i 102.20 ± 1.05
I-j 95.55 ± 1.02
1-DNJ 65.18 ± 1.04