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. 2022 May 13;5(6):400–412. doi: 10.1021/acsptsci.1c00264

Table 2. Average Pharmacokinetic Parameters of Pentarlandir UPPTA in Plasma in Each Animal Group.

condition/dosage Tmax (h) Cmax(μM) T1/2 (h) AUC0-t (μM·h) AUC0-∞ (μM·h)
fed, single dose/1000 mg/kg 3.40 ± 1.82 0.91 ± 0.35 3.90 ± 2.23 4.84 ± 1.92 6.73 ± 2.91
fasting, single dose/350 mg/kg 5.33 ± 0.82 0.69 ± 0.57 3.48 ± 2.44 2.39 ± 1.31 4.10 ± 1.73
fasting, single dose/750 mg/kg 2.60 ± 1.82 2.12 ± 0.65 2.58 ± 1.17 13.82 ± 7.61 13.94 ± 7.65
fasting, single dose/1000 mg/kg 3.71 ± 1.60 4.59 ± 1.36 2.74 ± 1.63 26.06 ± 9.58 30.16 ± 13.24
fasting, 14-day repeated dose/1000 mg/kg/day 4.83 ± 0.98 3.62 ± 1.74 6.01 ± 0.78 34.13 ± 11.39 36.73 ± 12.20