Table 2.

Potency and selectivity of ZED1227 against recombinant human transglutaminase isoenzymes.

ZED1227	hTG2	hTG1	hTG3	hTG6	hFXIII-A2
App. IC50	53 nM	24,863 nM	>50,000 nM	6,441 nM	>50,000 nM
Selectivity		469	>900	122	>900