Table 2.
Cytotoxic activity of the isolated compounds from Tylophora indica using MTT assays.
No. | Compounds | IC50 ± SD (μM) a | ||
---|---|---|---|---|
MCF-7 | HepG2 | HCT-116 | ||
1. | Tylophorine | 126.5 | 40.10 ± 2.94 | 142.20 ± 3.06 |
2. | Tylophorinicine | 50.71 ± 2.86 | 35.33 ± 2.97 | 75.55 |
3. | Tylophorinine | 31.96 ± 2.64 | 23.8 ± 3.02 | 86.95 ± 3.08 |
4. | Tylophorinine N-Oxide | ˃200 | 196.60 | ˃200 |
5. | Tylophorinidine | 6.45 ± 2.06 | 4.77 ± 2.11 | 20.08 ± 1.94 |
6. | Tylophorinidine-N-Oxide | 12.15 ± 1.81 | 15.31 ± 2.04 | 65.62 ± 2.24 |
7. | Septicine | ˃200 | ˃200 | ˃200 |
8. | Chlorogenic acid | 134.00 | 169.90 | ˃200 |
9. | Chlorogenic acid methyl ester | ˃200 | ˃200 | ˃200 |
10. | Cisplatin (Reference) | 5.70 ± 0.76 | 12.93 ± 0.91 | 14.42 ± 1.69 |
a IC50: Inhibitory concentration for 50%.