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Summary of data for FP1-24-2.A, structure of FP1-24-2. B, enzymatic profiling of FP1-24-2 against CK1γ family kinases. C, kinome tree representation of kinases with PoC <10 when FP1-24-2 was profiled at 1 μM versus 403 WT kinases. D, specific kinases (n = 14) with PoC <10 in kinome-wide profiling. E, Nanoluc-CK1γ2 NanoBRET curve and corresponding IC50 value for FP1-24-2. CK1γ, casein kinase 1γ; PoC, Percent of Control.
