Table 2.
Sensor | Ligand | Binding protein / module | Optical reporter | ΔF/F0 or FRET/BRET ratio | Kd or EC50 | Kinetics | In vivo application | Ref. |
---|---|---|---|---|---|---|---|---|
pmeLUC | ATP | No | Bioluminescence | ~8 | > 10 μM | N.D. | Mice | (Morciano et al., 2017) |
TANGO Assay | GPCR ligands | GPCRs | Reporter gene | >10 | ~ 1 nM | >8 h | N.D. | (Barnea et al., 2008) |
Sniffer cells | Adenosine, ATP, or ADP | A1R, P2X, or P2Y | Ca2+ sensor | ~1.5 (?) for Ado | 8 0μM (Ado) | N.D. | N.D. | (Yamashiro et al., 2017) |
ecATeam3.10 | ATP | Bacterial F0F1- ATP synthase | CFP/YFP | ~0.27 | ~11 mM | ~13–172 s (τon) | N.D. | (Conley et al., 2017) |
A2AR-based FlAsH | Adenosine | A2AR | CFP/FlAsH | ~0.1 | Similar to WT A2AR (?) | 66–88 ms (τon) | N.D. | (Hoffmann et al., 2005) |
P2X2-Cam | ATP | P2X2 | CFP/YFP | ~0.37 | ~14 μM | ~6 s (decay) | Zebrafish | (Richler et al., 2008) |
iATPSnFR | ATP | Bacterial F0F1- ATP synthase | cpSFGFP | ~1.0 | 350 μM | <5 s (τon), >1 s (τoff) | N.D. | (Lobas et al., 2019) |
N.D., not determined.