. 2022 Jun 19;17(7):1937–1950. doi: 10.1021/acschembio.2c00378

Table 1. Structure–Activity Relationship of the N-(3-Aminophenyl)acetamide Series of 3-Cyano-7-cyclopropylamino-pyrazolo[1,5-a]pyrimidines 1–7^a^,^b.

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In-cell target engagement of CSNK2A-nLuc in HEK293 cells. Data from ref (24).

Inhibition of MHV-nLuc replication in DBT cells. Values are the mean of three assays with range ± 15%.

Table 1. Structure–Activity Relationship of the N-(3-Aminophenyl)acetamide Series of 3-Cyano-7-cyclopropylamino-pyrazolo[1,5-a]pyrimidines 1–7a,b.