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. 2022 Jul 3;240:114576. doi: 10.1016/j.ejmech.2022.114576

Table 11.

Inhibition activity of isothiazolo [4,3-b]pyridine analogs against GAK.

Heterocyclic Scaffolds Kd (μM) Heterocyclic Scaffolds Kd (μM)
Image 58 0.052 Image 64 2
Image 59 0.77 Image 65 >30
Image 60 0.52 Image 66 0.041
Image 61 0.86 Image 67 >30
Image 62 0.4 Image 68 7.6
Image 63 >30 Image 69 3.2