Table 20.
Acetylene-substituted Anilinoquinazoline scaffolds showing inhibition to DENV.
| Heterocyclic Scaffolds | Inhibition Activity (EC50) (μM) | Heterocyclic Scaffolds | Inhibition Activity (EC50) (μM) |
|---|---|---|---|
![]() |
6.5 | ![]() |
9.0 |
![]() |
>10 | ![]() |
7.6 |
![]() |
>10 | ![]() |
5.0 |
![]() |
>10 | -- |
Acetylene-substituted Anilinoquinazoline scaffolds showing inhibition to DENV.
| Heterocyclic Scaffolds | Inhibition Activity (EC50) (μM) | Heterocyclic Scaffolds | Inhibition Activity (EC50) (μM) |
|---|---|---|---|
![]() |
6.5 | ![]() |
9.0 |
![]() |
>10 | ![]() |
7.6 |
![]() |
>10 | ![]() |
5.0 |
![]() |
>10 | -- |