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. 2022 Jul 3;240:114576. doi: 10.1016/j.ejmech.2022.114576

Table 24.

Inhibition activity of truncated benzothiazole-based heterocyclic scaffolds against DENV2 NS2B/NS3 protease.

Compound No. Heterocyclic Scaffolds IC50 (μM)
130 Image 138 26.95 ± 1.61
131 Image 139 4.38 ± 0.38
132 Image 140 5.97 ± 0.50
133 Image 141 6.39 ± 0.20
134 Image 142 4.86 ± 0.33