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. 2022 Jul 3;240:114576. doi: 10.1016/j.ejmech.2022.114576

Table 27.

Inhibition activity of various oxadiazole derivatives against the DENV2 RdRp.

Compound No. Heterocyclic Scaffolds IC50 (μM)
147 Image 155 2.2 ± 0.1
148 Image 156 6.0 ± 1.0
149 Image 157 3.5 ± 0.5
150 Image 158 4.8 ± 0.4
151 Image 159 4.0 ± 0.5
152 Image 160 11.0 ± 1.8
153 Image 161 9.1 ± 1.3