Table 27.
Inhibition activity of various oxadiazole derivatives against the DENV2 RdRp.
| Compound No. | Heterocyclic Scaffolds | IC50 (μM) |
|---|---|---|
| 147 | ![]() |
2.2 ± 0.1 |
| 148 | ![]() |
6.0 ± 1.0 |
| 149 | ![]() |
3.5 ± 0.5 |
| 150 | ![]() |
4.8 ± 0.4 |
| 151 | ![]() |
4.0 ± 0.5 |
| 152 | ![]() |
11.0 ± 1.8 |
| 153 | ![]() |
9.1 ± 1.3 |
Inhibition activity of various oxadiazole derivatives against the DENV2 RdRp.
| Compound No. | Heterocyclic Scaffolds | IC50 (μM) |
|---|---|---|
| 147 | ![]() |
2.2 ± 0.1 |
| 148 | ![]() |
6.0 ± 1.0 |
| 149 | ![]() |
3.5 ± 0.5 |
| 150 | ![]() |
4.8 ± 0.4 |
| 151 | ![]() |
4.0 ± 0.5 |
| 152 | ![]() |
11.0 ± 1.8 |
| 153 | ![]() |
9.1 ± 1.3 |