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. Author manuscript; available in PMC: 2022 Jul 7.
Published in final edited form as: Biochemistry. 2021 Jun 2;60(24):1933–1946. doi: 10.1021/acs.biochem.1c00215

Table 2.

Summary of Ki Values for HpAFLDAa

inhibitor Ki (nM) Ki* (nM)
(8R)-CF N/O N/O
(8R)-MTCF 560 ± 170 63 ± 4
(8R)-MT-2′d-CF N/O N/O
(8R)-PrT-2′d-CF 420 ± 140 N/O
(8R)-PhT-2′d-CF 850 ± 200 N/O
a

N/O means inhibition not observed.