The yields of synthesized products (4a–4u) using different derivatives of isatin, 3-aminopyrazole and isocyanide in the presence of CeCl3·7H2O catalysta.
Entry | Pyrazole | Isatin | Isocyanide | Product | Yield (%) |
---|---|---|---|---|---|
1 | 4a | 78 | |||
2 | 4b | 76 | |||
3 | 4c | 80 | |||
4 | 4d | 77 | |||
5 | 4e | 75 | |||
6 | 4f | 82 | |||
7 | 4g | 74 | |||
8 | 4h | 73 | |||
9 | 4i | 74 | |||
10 | 4j | 77 | |||
11 | 4k | 79 | |||
12 | 4l | 81 | |||
13 | 4m | 81 | |||
14 | 4n | 82 | |||
15 | 4o | 80 | |||
16 | 4p | 81 | |||
17 | 4q | 75 | |||
18 | 4r | 79 | |||
19 | 4s | 75 | |||
20 | 4t | 74 | |||
21 | 4u | 63 |
Isolated yield in the presence of CeCl3·7H2O catalyst (30 mol%).